{"id":2919,"date":"2018-07-18T10:53:26","date_gmt":"2018-07-18T10:53:26","guid":{"rendered":"https:\/\/adiccionsevilla.com\/?p=2919"},"modified":"2021-02-11T10:20:53","modified_gmt":"2021-02-11T10:20:53","slug":"la-proteina-para-curar-el-alcoholismo","status":"publish","type":"post","link":"https:\/\/forummontau.com\/sevilla\/la-proteina-para-curar-el-alcoholismo\/","title":{"rendered":"La prote\u00edna para curar el alcoholismo"},"content":{"rendered":"<p>El exceso de alcohol es malo para la salud. Y cuando este abuso se mantiene a lo largo del tiempo, el alcohol resulta simple y llanamente letal.<\/p>\n<p>Aunque es posible que el d\u00e9ficit de una prote\u00edna sea la responsable de que muchas personas no sean capaces de evitar el consumo y acaben desarrollando una adicci\u00f3n.<\/p>\n<h2>Prote\u00edna GAT-3 clave para explicar la adicci\u00f3n al alcoholismo<\/h2>\n<p>Un estudio muestra que los niveles bajos de la prote\u00edna GAT-3 en la am\u00edgdala son responsables de que el sistema de recompensa cerebral cambie sus \u2018preferencias\u2019 y priorice el alcohol sobre otras alternativas \u2018m\u00e1s saludables\u2019.<\/p>\n<p>Y lo que es m\u00e1s importante, que es muy posible que podamos contar con f\u00e1rmacos para corregir esta deficiencia y, as\u00ed, curar el alcoholismo.<\/p>\n<p>Como explica Markus Heilig, co-autor de esta investigaci\u00f3n publicada en la revista \u00ab<a href=\"http:\/\/www.sciencemag.org\/\">Science<\/a>\u00bb, \u00abtenemos que entender que\u00a0<strong>una de las caracter\u00edsticas principales de la adicci\u00f3n es que sabes que te va a hacer da\u00f1o, que potencialmente va a matarte, pero que sin embargo algo ha ido mal en el control motivacional y que sigues haci\u00e9ndolo<\/strong>\u00bb.<\/p>\n<p>En el estudio, los autores utilizaron un modelo animal \u2013ratas\u2013 que pod\u00eda obtener todo el alcohol que quisiera con el simple hecho de presionar una palanca. As\u00ed que los animales, dado que carec\u00edan de otra \u2018opci\u00f3n\u2019 para saciar su sed, se pasaban el d\u00eda borrachos.<\/p>\n<h2>Pero, \u00bfqu\u00e9 pasar\u00eda en caso de contar con una segunda alternativa? \u00bfSeguir\u00edan eligiendo el alcohol?<\/h2>\n<p>Pues para averiguarlo, los autores habilitaron una segunda palanca que, una vez presionada y a modo de recompensa, ofrec\u00eda agua azucarada. \u00bfY qu\u00e9 pas\u00f3? Pues que los animales decidieron dejar el alcohol y saciarse con el agua con az\u00facar, mucho m\u00e1s saludable. Pero no todos. El 15% de las ratas sigui\u00f3 optando por el alcohol, siendo este porcentaje similar al de los humanos con adicci\u00f3n al alcohol.<\/p>\n<p>Evidentemente, el objetivo del estudio no era conocer el porcentaje de ratas con problemas de alcoholismo, sino identificar los mecanismos subyacentes a los comportamientos adictivos.<\/p>\n<p>Y para ello, los autores analizaron la expresi\u00f3n de centenares de genes en cinco \u00e1reas del cerebro. Y lo que observaron es que la mayores diferencias en la expresi\u00f3n de genes entre ambos grupos de animales \u2013los devotos del agua azucarada y los partidarios del alcohol\u2013 se localizaron en la am\u00edgdala, regi\u00f3n cerebral que, entre otras muchas funciones, juega un papel primordial en las respuestas emocionales.<\/p>\n<p>Concretamente, los resultados mostraron\u00a0<strong>una expresi\u00f3n muy disminuida del gen \u2018GAT-3\u2019 en las am\u00edgdalas de los animales que optaban por seguir consumiendo alcohol<\/strong>. Un aspecto muy importante dado que este gen codifica la expresi\u00f3n de la prote\u00edna denominada \u2018transportador de GABA tipo 3\u2019 (GAT-3), responsable de mantener unos niveles adecuados del principal neurotransmisor inhibidor del sistema nervioso central \u2013el \u00e1cido \u03b3-aminobut\u00edrico (GABA)\u2013 en torno a las neuronas.<\/p>\n<p><strong>Esta carencia de prote\u00edna GAT-3, \u00bfest\u00e1 directamente implicada en la adicci\u00f3n al alcohol<\/strong> en estos animales? Pues para averiguarlo, los autores cogieron algunas de las ratas que hab\u00edan renunciado al alcohol y las manipularon gen\u00e9ticamente para que no pudieran expresar la prote\u00edna GAT-3, tras lo cual fueron reintroducidas en sus jaulas con las dos palancas \u2013agua azucarada y alcohol\u2013. Y de acuerdo con los resultados,<strong> la supresi\u00f3n de GAT-3 tuvo consecuencias catastr\u00f3ficas para la salud<\/strong> de los animales.<\/p>\n<p>Por tanto, la disminuci\u00f3n de los niveles de prote\u00edna GAT-3 juega un papel determinante en el desarrollo de la adicci\u00f3n al alcohol en ratas. Pero: \u00bfsucede lo mismo en los humanos? Pues s\u00ed.<\/p>\n<h2>La concentraci\u00f3n de esta prote\u00edna en la am\u00edgdala es inferior en personas con alcoholismo<\/h2>\n<p>Los autores analizaron los niveles de GAT-3 en los tejidos cerebrales de pacientes con adicci\u00f3n al alcohol ya fallecidos. Y de acuerdo con los resultados, la concentraci\u00f3n de esta prote\u00edna en la am\u00edgdala fue muy inferior a la observada en los cerebros de personas que, igualmente fallecidas, no hab\u00edan desarrollado esta adicci\u00f3n.<\/p>\n<p>En este contexto, ya hay disponible un f\u00e1rmaco que, denominado \u2018baclofeno\u2019 y utilizado desde hace ya muchos a\u00f1os para aliviar la tensi\u00f3n muscular en algunas enfermedades neurol\u00f3gicas, ha mostrado un gran potencial en el tratamiento de la dependencia al alcohol.<\/p>\n<p>Sin embargo, el mecanismo por el que se explicaba esta eficacia frente al alcoholismo permanec\u00eda desconocida. Hasta ahora.<\/p>\n<p>Como concluye Markus Heilig, \u00abuna de las cosas que hace el baclofeno es suprimir la liberaci\u00f3n de GABA.<\/p>\n<p>En la actualidad estamos trabajando con una compa\u00f1\u00eda farmac\u00e9utica para\u00a0<strong>tratar de desarrollar una mol\u00e9cula de segunda generaci\u00f3n como posible f\u00e1rmaco candidato para el tratamiento del alcoholismo a trav\u00e9s de la actuaci\u00f3n dirigida sobre esta v\u00eda de se\u00f1alizaci\u00f3n<\/strong>\u00bb.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>El exceso de alcohol es malo para la salud. Y cuando este abuso se mantiene a lo largo del tiempo, el alcohol resulta simple y llanamente letal. Aunque es posible que el d\u00e9ficit de una prote\u00edna sea la responsable de que muchas personas no sean capaces de evitar el consumo y acaben desarrollando una adicci\u00f3n. [&hellip;]<\/p>\n","protected":false},"author":8,"featured_media":2921,"comment_status":"closed","ping_status":"closed","sticky":false,"template":"","format":"standard","meta":{"ocean_post_layout":"","ocean_both_sidebars_style":"","ocean_both_sidebars_content_width":0,"ocean_both_sidebars_sidebars_width":0,"ocean_sidebar":"0","ocean_second_sidebar":"0","ocean_disable_margins":"enable","ocean_add_body_class":"","ocean_shortcode_before_top_bar":"","ocean_shortcode_after_top_bar":"","ocean_shortcode_before_header":"","ocean_shortcode_after_header":"","ocean_has_shortcode":"","ocean_shortcode_after_title":"","ocean_shortcode_before_footer_widgets":"","ocean_shortcode_after_footer_widgets":"","ocean_shortcode_before_footer_bottom":"","ocean_shortcode_after_footer_bottom":"","ocean_display_top_bar":"default","ocean_display_header":"default","ocean_header_style":"","ocean_center_header_left_menu":"0","ocean_custom_header_template":"0","ocean_custom_logo":0,"ocean_custom_retina_logo":0,"ocean_custom_logo_max_width":0,"ocean_custom_logo_tablet_max_width":0,"ocean_custom_logo_mobile_max_width":0,"ocean_custom_logo_max_height":0,"ocean_custom_logo_tablet_max_height":0,"ocean_custom_logo_mobile_max_height":0,"ocean_header_custom_menu":"0","ocean_menu_typo_font_family":"0","ocean_menu_typo_font_subset":"","ocean_menu_typo_font_size":0,"ocean_menu_typo_font_size_tablet":0,"ocean_menu_typo_font_size_mobile":0,"ocean_menu_typo_font_size_unit":"px","ocean_menu_typo_font_weight":"","ocean_menu_typo_font_weight_tablet":"","ocean_menu_typo_font_weight_mobile":"","ocean_menu_typo_transform":"","ocean_menu_typo_transform_tablet":"","ocean_menu_typo_transform_mobile":"","ocean_menu_typo_line_height":0,"ocean_menu_typo_line_height_tablet":0,"ocean_menu_typo_line_height_mobile":0,"ocean_menu_typo_line_height_unit":"","ocean_menu_typo_spacing":0,"ocean_menu_typo_spacing_tablet":0,"ocean_menu_typo_spacing_mobile":0,"ocean_menu_typo_spacing_unit":"","ocean_menu_link_color":"","ocean_menu_link_color_hover":"","ocean_menu_link_color_active":"","ocean_menu_link_background":"","ocean_menu_link_hover_background":"","ocean_menu_link_active_background":"","ocean_menu_social_links_bg":"","ocean_menu_social_hover_links_bg":"","ocean_menu_social_links_color":"","ocean_menu_social_hover_links_color":"","ocean_disable_title":"default","ocean_disable_heading":"default","ocean_post_title":"","ocean_post_subheading":"","ocean_post_title_style":"","ocean_post_title_background_color":"","ocean_post_title_background":0,"ocean_post_title_bg_image_position":"","ocean_post_title_bg_image_attachment":"","ocean_post_title_bg_image_repeat":"","ocean_post_title_bg_image_size":"","ocean_post_title_height":0,"ocean_post_title_bg_overlay":0.5,"ocean_post_title_bg_overlay_color":"","ocean_disable_breadcrumbs":"default","ocean_breadcrumbs_color":"","ocean_breadcrumbs_separator_color":"","ocean_breadcrumbs_links_color":"","ocean_breadcrumbs_links_hover_color":"","ocean_display_footer_widgets":"default","ocean_display_footer_bottom":"default","ocean_custom_footer_template":"0","ocean_post_oembed":"","ocean_post_self_hosted_media":"","ocean_post_video_embed":"","ocean_link_format":"","ocean_link_format_target":"self","ocean_quote_format":"","ocean_quote_format_link":"post","ocean_gallery_link_images":"off","ocean_gallery_id":[],"footnotes":""},"categories":[2,3,43,12],"tags":[42,41],"class_list":["post-2919","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-adicciones","category-alcohol","category-gat-3","category-tratamientos","tag-adicciones-sevilla","tag-forum-sevilla","entry","has-media"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.6 - 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